Compile Data Set for Download or QSAR
maximum 50k data
Found 14 of ki data for polymerid = 4005,10082
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
University Of Delhi

Curated by ChEMBL
LigandPNGBDBM50276305(CHEMBL4127220)
Affinity DataKi:  841nMAssay Description:Inhibition of Plasmodium falciparum Plm4 using synthetic substrate pretreated for 5 mins followed by substrate addition measured immediately by spect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
University Of Delhi

Curated by ChEMBL
LigandPNGBDBM50276293(CHEMBL4125845)
Affinity DataKi:  1.98E+3nMAssay Description:Inhibition of Plasmodium falciparum Plm4 using synthetic substrate pretreated for 5 mins followed by substrate addition measured immediately by spect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
University Of Delhi

Curated by ChEMBL
LigandPNGBDBM50276301(CHEMBL4128581)
Affinity DataKi:  3.35E+3nMAssay Description:Inhibition of Plasmodium falciparum Plm4 using synthetic substrate pretreated for 5 mins followed by substrate addition measured immediately by spect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32387(phenyl-substituted sulfonamides, 6d)
Affinity DataKi:  7.50E+3nM ΔG°:  -6.94kcal/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32388(phenyl-substituted sulfonamides, 6e)
Affinity DataKi:  7.50E+3nM ΔG°:  -6.94kcal/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32385(phenyl-substituted sulfonamides, 6b)
Affinity DataKi:  1.70E+4nM ΔG°:  -6.46kcal/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32389(phenyl-substituted sulfonamides, 6f)
Affinity DataKi:  2.00E+4nM ΔG°:  -6.36kcal/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32384(phenyl-substituted sulfonamides, 6a)
Affinity DataKi:  3.60E+4nM ΔG°:  -6.02kcal/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32386(phenyl-substituted sulfonamides, 6c)
Affinity DataKi:  4.20E+4nM ΔG°:  -5.93kcal/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32391(iso-butyl-substituted sulfonamide, 9b)
Affinity DataKi:  5.60E+4nM ΔG°:  -5.80kcal/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32393(carboxamide, 12b)
Affinity DataKi:  5.60E+4nM ΔG°:  -5.80kcal/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32390(iso-butyl-substituted sulfonamide, 9a)
Affinity DataKi:  8.70E+4nM ΔG°:  -5.50kcal/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32392(carboxamide, 12a)
Affinity DataKi:  9.80E+4nM ΔG°:  -5.46kcal/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32394(carboxamide, 12c)
Affinity DataKi:  1.70E+5nM ΔG°:  -5.14kcal/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed